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Tamoxifen citrate is one of the most widely used medicines in bodybuilding, but most often it is used as a protection, and not as an active ingredient. Most of those who are familiar with doping in bodybuilding associate it with anabolic steroids, but tamoxifen does not belong to this category. Basically known as nolvadex, or nolva, tamoxifen is most commonly used in bodybuilding by those who use anabolic steroids for two purposes: during the course to prevent side effects, and even more often during PCT (therapy after an anabolic steroids course). Basically, tamoxifen is well tolerated, this applies to both men and women, but the ladies mostly use it in much smaller doses and do it for the sake of its active, not protective effect.
Tamoxifen was first synthesized in 1962 in an attempt to create a contraceptive pill taken the day after intercourse. His tests showed that he did not give the desired effect, but soon found other valuable qualities. It was understood that it was estrogen that is a problem hormone in those who suffer from breast cancer. In tamoxifen, a property was found to block the interaction of estrogen with its receptors. At the same time the level of estrogen in the body did not decrease, and it was very valuable.
While the benefits of tamoxifen in combating breast cancer have been proven, other useful properties have been found. Increasing estrogen is a bodybuilding problem for many who use anabolic steroids. This is due to the effect of their aromatization. Tamoxifen allows to solve problems in bodybuilders, associated with an increase in the level of estrogen.
Properties and Functions of Tamoxifen citrate
Tamoxifen Citrate is a SURM with the properties of both the agonist and the antagonist of estrogen. As an antiestrogen, Nolvadex functions by binding to estrogen receptors at the site of estrogen. This binding prevents the hormone estrogen from carrying out its actions in certain parts of the body, which is why it is extremely useful for breast cancer patients. Many forms of breast cancer actually “eat” estrogen when it is attached to the breast receptors. Preventing such attachment of receptors also protects anabolic steroids users from gynecomastia, which can be caused by aromatizing to a certain extent anabolic steroids, such as Testosterone, Dianabol, Nandrolone and Boldenone.
Although the drug is primarily considered an antiestrogen, Nolvadex has the ability to act as an estrogen, especially in the liver. What gives an advantage, since such estrogenic activity in the liver is associated with more healthy levels of cholesterol. For users of steroids, this can be very useful, since many anabolic steroids have a negative effect on cholesterol. More details on this will be discussed in the section “The Action of Nolvadex.”
Being primarily an antiestrogen, Nolvadex also has strong testosterone stimulant properties. Nolvadex has the ability to block negative adverse effects of estrogen on the hypothalamus and pituitary gland. As a result, the release of Luteinizing Hormone (LH) and Follicle-stimulating Hormone (FSH) increases. Both hormones are of great importance for the production of natural testosterone. Without LH and FSH, especially without LH, the production of natural testosterone is impossible.
Side effects of Tamoxifen citrate
Side effects are possible with the reception of Nolvadex, but this SORM is well tolerated by both men and women. Possible side effects, however, are very rare. Most men will not have the first problem. Side effects from Nolvadex most often occur in women, but even then they will not be common to all. Possible side effects from Nolvadex include:
- Vaginal itching, bleeding, discharge or discomfort
- Stomach upset
The above effects are the most common. Other possible side effects of Nolvadex, although less frequent than the above, include:
- Reducing the number of leukocytes
- Changes in the endometrium
- Increased triglyceride levels
- Pulmonary embolism
When we talk about the side effects of Nolvadex, then that’s really all. Undoubtedly, some of these effects sound unpleasant, but again, most of them are quite rare. As a last comment, pregnant women or those who can become pregnant should not take Nolvadex under any pretext. Such a technique can be very dangerous for an evolving child.
Tamoxifen citrate for men. Description, effects from admission
- Tamoxifen during the course fights with 1 sign of gynecomastia;
- The blockade of estrogen;
- Has a low price;
- Effectively affects the state of the lipid profile;
- Rapid assimilation, which in turn is important for the initial occurrence of gynecomastia;
- There is an anti-catabolic effect (protects meat);
- No. 1 for Post-Course Therapy (with the exception of Nandrolones and Trenbolones).
Tamoxifen citrate on the course
Do not confuse the use of Tamoxifen using a variety of aromatase inhibitors. Such drugs block the conversion to estrogens, Tamoxifen, in turn, matches the estrogen receptor, becomes in their place, so they are not able to lead to gino and damage the course. Such guarantees absolute protection against estrogenic pobochek, such as a drop in libido, high irritability, fluid accumulation, lethargy, gynecomastia, and others.
One of the most well-known uses is tamoxifen for gynecomastia. If you feel that the nipples are ache a little or it itch, in this case the timely taking of a small dose of Nolvadex will solve the problem. For the sake of justice, it must be emphasized that all types of this type of drugs can only help in the first stages of gynecomastia. Any effective steroidal course of anabolic drugs can not exist without optimal post-course therapy.
Tamoxifen for increasing testosterone takes place after each course of anabolic steroids, excluding courses with Nandrolone, and Tren.
The advantage of this category of pharma is incredibly useful during post-course therapy, when the values â€‹â€‹of Testosterone decrease, due to the stopping of anabolic intake, while female hormones still remain at a high level and do not allow the body to restore the hormonal background.
Tamoxifen citrate after the course
The main role of Tamox’s play is played precisely after the conducted courses and is necessary for PKT. In this case, this is an unequivocal necessity. After the abolition of steroids, the level of Testosterone, as well as dihydrotestosterone, is extremely reduced. The body needs to be renewed, while doing this against the background of a huge volume of female elements is hardly feasible. What to do? – Take Tamoxifen.
A large estrogen index contributes to the loss of results obtained during the course of application of drugs sport pharma. Nolva for a while will block estrogens, because of this the body will have the opportunity to resume itself well.
It should be noted that it is also necessary to promptly “press” cortisol, which destroys together with female estrogens the obtained muscles in PKT. Maple and Tamoxifen – with their help inhibited catabolism, as well as loss of muscle fibers. Tamox (20 mg) plus Maple (20 – 40 micrograms) per day. Clenbuterol gives a small bonus – you can pile more on the plate and not be afraid that you swim with fat in the period of PBC.
Tamoxifen citrate – Feedback
Nolvadex is an example of a very effective antiestrogen, moreover, inexpensive. Tamox in sports is known no less than in the general medical environment. For the most part, thanks to the cheapness, he is chosen instead of Clomid. Tamoxifen – reviews of men on the drug are uniquely positive. Blocking the work of female hormones allows athletes to lose weight, to maintain stiffness and muscle tone.
The drug is used after all types of steroid courses. In general terms – it is the most important restorative preparation among the kit for each chemist.
Antiestrogens are required absolutely for all male athletes who consume steroid drugs. In case, for individual reasons, Tamoxifen citrate does not suit you, you can buy a substitute of Tamoxifen, for example, Clomid. Tamox in bodybuilding is in demand not less than steroid preparations.
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